… Cyproheptadine has been chosen by our group as the starting point of a search for … of the
cyproheptadine analogues 2f—j and 3b at the 5-HT2A, 5-HT23 and 5HTZC receptors correlate …

… with 5-HT2A, 5HT2B, and 5-HT2C subpopulations [1]. Depending on the … of parallel
structure-activity relationships between two series of … Several cyproheptadine analogs with altered …

… The discrimination of 5-HT2A, 5-HT2C and 5-HT2C receptors … studies focused on analogs
of the 5-HT2A receptor antagonist … quantitative structure-activity relationships (QSAR) and to …

… at 5-HT2B receptors, a series of DOX analogues was analyzed … structure-activity relationships
of risperidone antagonism at … 5-HT1D, 5-HT2A, 5-HT2C, and sigma-1 receptors.Fen clearly …

… This receptor family is comprised of three subtypes: 5HT2A, 5-HT2B, and 5-HT2C receptors.
-… Among these, mutagenesis, imaging, and structure-activity relationship (SAR) formulation …

… , we choose ketanserin and cyproheptadine to represent the … (67-70) Structure–activity
relationship (SAR) studies on … study, we designed series of sorafenib analogues to assess the …

… points, each group of tricyclic 2-aminotetralin analogues was … previously discussed [40]
structure-activity relationships: (a) … , namely 5-HT2A, 5-HT2B and 5-HT2C receptors. Like the 5-…

… Structureactivity relationships (SAR) of these ligands will … 5-HT receptor subtypes, except
5-HT2A (30-fold), 5-HT2B (50-… were also selective over 5-HT2C and 5-HT6 receptors, and to a …

… re-uptake, but without affinity to histamine and muscarinic receptors. On the other hand, … HT
2 receptors, since these effects were completely antagonized by cyproheptadine in the group …

… Tested compounds are claimed to be selective over a number of receptors such as serotonin
5-HT1A, 5HT2A, 5-HT2B, 5-HT2C, 5-HT3, 5-HT4, and 5-… = Structure activity relationships …